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第十三章 医薬関連発明 - 台湾知的財産権情報サイト

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Contents

1.
2.
3.
4. 2013 2 13 38
5. 3 1 1 2 oe 0 i
6. R
7. SR 1
8. kal TH
9. HH k 1 ii 2 13 25 2013 i Y 2 2
10. 2 13 6 lt
11. 1 B X B B X
12. 2 2 1 1 3 3 2 13 2
13. MM OO 2 13 3 2013 2013
14. 3 1 1 1 6
15. 1 ower alkyl 0 CT CHs E
16. 2 5 2 4 Y
17. 2 2 1 2 1 1 X 2 C 3 4 C
18. 3 a Met Ala Ala 2 13 16 b HIV Met Ala Ala A DNA DNA A A
19. 26 2 3 3 1 REE SEE
20. A
21. 4 1 R R N OH 2 R R N N R OR R Rs Y 2 13 43 2013 1 2
22. NR 24 2 4 2 OG MH
23. 5 3 2 5 3 2 1 1 2 13 37 2013
24. A MR A
25. 1
26. 1 ss lt 2 13 13 2013
27. 1 1a O N N 2013 2 13 34 1b O 2 1 N N N 1b 1a 2 2a H N C H4 SO NHR 2b HLN C H4 SO gt NHCONHR 2 25
28. enantiomer racemic mixture 2013 2 13 28 RM CS
29. kit package combination A X A X A A X X
30. 2013 RM 2 0 5 0mg kg 3 2 13 22 A 5 0 10 0mg kg 2
31. XX X IR Raman NMR DTA TGA DSC X A A 2 13 21 2013 4 2 1 2 ND NN
32. NO NN Y 2 13 2013 2013 RA
33. ee US 0 3 1 1 1 1 i 2 13 10
34. 5 2 1 2 1 1 element sub sets sub ranges Ne NSH X Ri COOH
35. 2 3 3 E
36. X Y 0 A NG
37. 2 13 17 2013 A A A A A HIV
38. Gi Gov 2 13 27 2013
39. A 5 NSH oO 0 MM HIV A ON
40. 2 H H HH Bi cimetidine ranitidine famotidine roxatidine acetate H H
41. NAO i ENA NH A A NC A A B A B
42. 5 8 jl OT 0 MN 22 Es 5 3 1 1 2 position isomers CH 2
43. MR 2 2 2 2 1 24 24
44. 5 3 3
45. 6 2 2 1 2 A B
46. RI A UVA UVB A UVA UVB
47. 2 13 7 2013 2013 0 8 0 E 2
48. 2 13 36 RB SCO NKK R 1
49. 7 31 7 1 7 1 1 alternatives nature
50. geometrical isomers homologues 5 3 1 2 enantiomer 0 i racemic mixture
51. 2 13 11 2013
52. a 9 I i A NN
53. 0 R X R XX 2013 2 13 18 D X R
54. 2 2013 D 1 2 IL X A 1
55. X 2 X NG Ni EHH MRD
56. UVA UVB 2 2 1 3
57. 2 2 1 2 1
58. analsesic decongsestant 1 2 2 13 39 2013 2013
59. A B C A B C A B C X 1 1 2 X X
60. Xe dissolve Xe 2 Xe Xe MR 2 13 8 2 2 2 1
61. 1 ed A RE A A 5 2 1 1 A Re y
62. on NM 3 1 3 1 1 X X X
63. 2013 2 13 14 A A B C 1 X
64. 5 3 1 3 LU 8 2 ti aie am A 8
65. 1 77 2 13 1 2 SRA 2 13 1 2 SR 2 lh 1 2 13 1 a 2 13 1 2 en 2 13 2 2 2 13 2 2 2 i 2 13 2 2 2 1 2 13 2 2 2 1 1 kk 2 13 2 2 2 1 2 kk 2 13 5 2 2 1 3 i 2 13 7 2 2 2 I 2 13 9 2 13 9 3 ON 2 13 9 93U KN 2 13 9 3 EE 2 13 10 3 1 1 1 1 kk 2 13 10 3 1 1 1 2 IIIIIIIIIEILIILILIL kk 2 13 11 3 15113 ER 2 13 11 3 1 1 2 tka a 2 13 12 3 1 1 3 kt 2 13 12 3 1 2 Ek 2 13 13 3 1 3 kk 2 13 14 4620800088k 2 13 19 0 PIE 2 13 19 PS BE MOD ME mA 2 13 20 2 00ORS ARE0000338000S22 RS28R238E22HR38 8 2 13 21 4 2 1 1 iii 2 13 21 4 2 1 2
66. A B C D E A Ci Cijp C gt Cj Ca Cij O N 1 3 Cs C B Ci C Co gt C Co C Cs C C O S N 1 4 Cs C 2013 2 13 42 Bs 526 D B C4 C E A B C D E
67. pH
68. 1 G 4 2 13 31 2013 2013
69. 1 B I 4 2 1 2 1 2 13 23 2013 2013 X X X OO OO X
70. a 1 element b 1 component
71. 2 13 26 22 1 22 1 4 2 4 1 0 2 I 1 is
72. 2 5 5 1 5 2 5 2 1 1 1
73. 24 2 X 2 DO 1 6
74. 26 1 3 1 1 2 13 9 2013 2013 RA NR MO 0 amount of oo
75. 1 SCH R N C CH z NG Rr ZZ N C SCHs 2 13 41 2013
76. RAR 4 2 1 3
77. A A 4 D X 1 R O C HL CH CH3 COOH R C Co 1 3 XX X R X
78. X 2 X 1 i MM XX XX X 0 X A B C
79. 26I 2 4 2 13 20 4 2 1 2 4 1 4 2 1 1
80. 2 1 Ri R gt R 3
81. NR NN 24 2 2 2 1 1
82. B A X X B E 2 13 19 2013 2013 Swiss type claim A X A X A
83. Xe 1 2 13 4 Xe dissolve Xe NIR OB NN
84. 5 2 2 1 1 1 1 5 2 2 1 2 A Z A
85. X R XX 4 4 1 A
86. 7 2 1 2013 2 13 44
87. i oo microarray I
88. 5 3 2 2 ii
89. 1 S 0 lu mu ll ll 2 13 24 4 2 2 2 4 2 4 2 3 Markush type
90. IL X TL X 1 1 OH R HH N N 9 IL X R1 R2 C1 6 MNO L X 5 ILX 1 IL X
91. X Gnstruction X Y 2 13 32 5 3 5 3 1 Ds
92. A A A A i NN A A A HIV A homology HIV A
93. R CHbCHLCH R2 gt C1 SO3sH CH3 0 X Phenyl R gt COOH CHoCH2CH 2 Nh R COOH NH CI SO H CH 2 13 29 CH CH CH Ri COOH CHzCH2CH3 Ri R gt C
94. 1 Xe 3 1
95. 5 3 1 4 0 002 3 3a 3b ME 4b 4b Ee 2013
96. 2 13 15 2013 2013 A 5 A A A RNN RS MR i A
97. 5 2 13 1 1 I 2013 2013 2 1 2 3 2 1 3 1
98. i 2 13 22 4 2 1 3 ki 2 13 23 422 Eo Rk 2 13 25 4 2 3 kk 2 13 25 2 KK 2 13 27 2 13 1 5 2 13 27 S680 0S EEE RT 13 5 1 kt 2 13 27 SS 2 13 27 521 NN 2 13 27 5 2 1 1 i 2 13 28 5912 6 RENNN 2 2 13 29 522 2 13 30 5 2 2 1 Hi 2 13 30 2 2 1 1 1 2 13 30 5 2 2 1 2 2 13 30 5 2 3 iki 2 13 31 5 2 4 2 13 32 223 2 13 33 3A kk Rk 2 13 33 5 3 1 1 kkk 2 13 33 5 3 1 2 kk 2 13 33 5 3 1 3 kkk 2 1
99. 0 8 pH 3 1 1 3 3 1 1 1 3 2013 2 13 12 3 1 2
100. 2 2b 3 3a CONHCH CH H C CH 3b CONHCH H C CH 3a 35 2 13 35 2013 30 90 ul 4 3b 4a O No CH O OCH ul O N_o _ P CH O SCH NO 4b NO 4a SCH OCH
101. 2 b 2 13 40 1 7 1 2 2 4
102. 2 13 33 2013 2
103. 3 1 1 1 2 1 3 1 1 1 3 SW A
104. A Y A 5 0 10 0 mg kg 2 2 0 5 0mg kg 3 A Y X X A
105. X A Z A 2 13 30 5 2 3 A A
106. X
107. mM X a 1 OO 2 2 A
108. b Gj 2 1 b
109. a X X A B C A B C A B C X X A B C X
110. 3 34 5 3 1 4 kkk 2 13 36 5 3 2 kk 2 13 37 5 3 2 1 2 13 37 3 2 2 2 13 38 5 3 3 ikki 2 13 38 6 ua uaau uu uaa autuuuuuaaaaaeeeeeeea 2 13 39 SR 2 13 40 7 1 lk 2 13 40 RNN eeh22080N80RDBTS2 5 2 13 40 7 1 2 kk 2 13 41 7 2 2 13 44 2 13 1 lll
111. A B 3 3 2 2 2 2 synergistic effecD 2
112. HzCH2CH Ri R COOH 2013 2013 5 2 2 1 1 5 2 2 1

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